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Search Result

Search Results for " orphan g-protein coupled receptor "

Targets

GPR

23

Compounds

6

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T23204 PSN 375963 PSN 375963 hydrochloride GPR
PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.
T5422 CID 1375606 CID-1375606,CID1375606 Others
CID 1375606 is a surrogate agonist of orphan G protein-coupled receptor GPR27. characterized by a high level of conservation among vertebrates and a predominant expression in the central nervous system.
TP2073L BigLEN (mouse) acetate BigLEN (mouse) acetate (501036-69-7 Free base) GPR
BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.
T60199 NCRW0005-F05 GPR
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 value of 0.21 μM. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson's disease [1].
TP1982L Neuropeptide S (Rat) acetate Neuropeptide Y Receptor
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor. Neuropeptide S (Rat) acetate can be used for the research of nervous system disease [1].
T19700 IBC 293 IBC293,IBC-293 GPR
IBC 293 is selective for GPR109B over niacin receptor GPR109A. IBC 293 is a highly selective agonist for GPR109B, a human orphan G-protein-coupled receptor expressed in adipocytes.
T70771 PSB-1737
PSB-1737 is a Potent Agonists of the Orphan G Protein-Coupled Receptor GPR17 (EC50 270 nM).
T68805 PSB-1584
PSB-1584 is a Potent Agonist of the Orphan G Protein-Coupled Receptor 84 (GPR84). GPR84, a Gi protein-coupled receptor that is activated by medium-chain (hydroxy)fatty acids, appears to play an important role in inflamma...
T83547 (Des-Bromo)-Neuropeptide B (1-23) (human)
'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM for GPR8 (NPBW2) respectively [1].
T75962 Urotensin II, mouse acetate
Urotensin II, mouse acetate, serves as an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR and acts as a potent vasoconstrictor. Its physiological function extends to the central nervous system [...
T68247 PSB-KD107
PSB-KD107 is an agonist of the Cannabinoid-Activated Orphan G‑Protein-Coupled Receptor GPR18. PSB-KD107 displayed significantly higher potency and efficacy than THC, determined in a GPR18-dependent β-arrestin recruitment...
T75961 Urotensin II, mouse TFA
Urotensin II, mouse TFA, an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR, serves as a potent vasoconstrictor. It plays a significant physiological role within the central nervous system [1].
T83743 VPM-p15 TFA T1V/F3Phe(4-Me)
VPM-p15, a synthetic peptide agonist targeting the adhesion G protein-coupled receptor (GPCR) G2 (ADGRG2)—an orphan GPCR implicated in male infertility—facilitates cAMP accumulation in HEK293 cells expressing human ADGRG...
T81683 Neuromedin S (human)
Neuromedin S (human) is a 33-amino acid neuropeptide identified as an endogenous ligand for the orphan G-protein coupled receptor (GPCR) FM-4/TGR-1, acting on the neuromedin U (NMU) receptor 2 (NMUR2) to regulate body we...
T75784 Apelin-36(rat, mouse) TFA
Apelin-36(rat, mouse) TFA, an endogenous agonist for the orphan G protein-coupled receptor APJ, exhibits a strong affinity for APJ receptors with an IC 50 of 5.4 nM and effectively inhibits cAMP production with an EC 50 ...
T69612 PSB-KD477
PSB-KD477 is an Agonist of the Cannabinoid-Activated Orphan G-Protein-Coupled Receptor GPR18. PSB-KD477 displayed significantly higher potency and efficacy than THC, determined in a GPR18-dependent β-arrestin recruitment...
T75785 Apelin-17(human, bovine) TFA
Apelin-17(human, bovine) TFA is an endogenous agonist of the orphan G protein-coupled receptor APJ. This compound demonstrates affinity for human APJ receptors on HEK 293 cells, evidenced by a pIC50 value of 9.02. Additi...
T75925 Orexin B, rat, mouse TFA
Orexin B, rat, mouse (Rat orexin B) TFA, an endogenous agonist for orexin receptors, binds to and activates the closely related orphan G protein-coupled receptors OX1-R and OX2-R. This compound is instrumental in stimula...
T35794 Kisspeptin-54 (human) (trifluoroacetate salt)
Kisspeptin-54 is a peptide ligand of the orphan G protein-coupled receptor GPR54 (Kis = 1.81 and 1.45 nM for rat and human receptors, respectively).1 It is a 54 amino acid peptide encoded by the metastasis suppressor gen...
T75783 Apelin-36(human) TFA
Apelin-36(human) TFA, an endogenous agonist of the orphan G protein-coupled receptor APJ, exhibits a potent EC50 of 20 nM and high affinity (pIC5 50 = 8.61) for human APJ receptors in HEK 293 cells. It is involved in sig...
T83926 S-Geranylgeranyl-L-glutathione GGG
S-Geranylgeranyl-L-glutathione acts as a ligand for the orphan G protein-coupled receptor (GPCR) P2RY8, displaying selective affinity by inducing internalization of P2RY8 in preference to the sphingosine-1-phosphate rece...
T37187 D-erythro/L-threo Lysosphingomyelin (d18:1) D-erythro/L-threo Lysosphingomyelin (d18:1)
Lysosphingomyelin is an endogenous bioactive sphingolipid and a constituent of lipoproteins.1,2It is produced by the removal of the acyl group from sphingomyelin by a deacylase and acts as a precursor in the biosynthesis...
T35597 Neuromedin U-23 (rat) (trifluoroacetate salt)
Neuromedin U-23 (NMU-23) is a neuropeptide involved in diverse biological processes, including smooth muscle contraction, energy homeostasis, and nociception.1It is an agonist of neuromedin-U receptor 1 (NMUR1; EC50= 0.1...

Recombinant Proteins

Species：
Human (4)
Cynomolgus (1)
Mouse (1)
Expression System：
HEK293 Cells (6)
Tag：
(2)
C-His (2)
C-His-Avi (2)
Cat No. Product Name Species Expression System
TMPK-00528 GPRC5D Protein-VLP, Cynomolgus, Recombinant Cynomolgus HEK293 Cells
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP...
TMPK-01193 GPRC5D Protein-VLP, Mouse, Recombinant Mouse HEK293 Cells
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP...
TMPY-04270 GPR133 Protein, Human, Recombinant (His) Human HEK293 Cells
ADGRD1 (Adhesion G Protein-Coupled Receptor D1, also known as GPR133) is a Protein Coding gene. 4 alternatively spliced human isoforms have been reported. ADGRD1, an orphan member of the adhesion family of G-protein-coup...
TMPY-02717 GPR37 Protein, Human, Recombinant (His) Human HEK293 Cells
GPR37 (cathepsin Z) is an orphan receptor that belongs to the G-protein coupled receptor 1 family. G protein-coupled receptors are a large protein family comprised of transmembrane receptors that sense molecules outside ...
TMPK-01411 Peptide Ready HLA-G&B2M Monomer Protein, Human, MHC (His & Avi), Biotinylated Human HEK293 Cells
Peptide Ready HLA-G&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-G. Peptide ready MHC molecules comprising human HLA alleles and B2M, which can b...
TMPK-01418 Peptide Ready HLA-G&B2M Monomer Protein, Human, MHC (His & Avi) Human HEK293 Cells
Peptide Ready HLA-G&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-G. Peptide ready MHC molecules comprising human HLA alleles and B2M, which can b...
Cat No. Product Name
L2610 Neurotransmitter Receptor Compound Library

1513 compounds
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；

Libraries

Neurotransmitter Receptor Compound Library
L2610
Compounds: 1513
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